MAP3K1
KINASE INFORMATION
Kinase Name
mitogen-activated protein kinase kinase kinase 1
Entrez Gene Symbol
MAP3K1
Entrez Gene ID
4214
Aliases
MAP3K1; MAPKKK1; MEKK; MEKK1; MEKK1/MAP3K1
Kinase Group
STE
Species
Human
PROTEIN INFORMATION
Accession #
NP_005912.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.65
Panel
Delta Set CE; Delta Set I; Delta Set M; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
4400 nM
Staurosporine
350 nM