MAP4K5
KINASE INFORMATION
Kinase Name
mitogen-activated protein kinase kinase kinase kinase 5
Entrez Gene Symbol
MAP4K5
Entrez Gene ID
11183
Aliases
GCKR; KHS; KHS1; MAP4K5; MAPKKKK5
Kinase Group
STE
Species
Human
PROTEIN INFORMATION
Accession #
NP_006566.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.75
Panel
Delta Set CA; Delta Set CE; Delta Set M; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
43 nM
Dasatinib
45 nM
Sunitinib
41 nM