MAST1
KINASE INFORMATION
Kinase Name
microtubule associated serine/threonine kinase 1
Entrez Gene Symbol
MAST1
Entrez Gene ID
22983
Aliases
KIAA0973; MAST1; SAST; SAST170
Kinase Group
AGC
Species
Human
PROTEIN INFORMATION
Accession #
NP_055790.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.5
Panel
Delta Set CA; Delta Set CE; Delta Set I; Delta Set M; Delta Set RB; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
19 nM
Staurosporine
150 nM
Sunitinib
200 nM