MELK
KINASE INFORMATION
Kinase Name
maternal embryonic leucine zipper kinase
Entrez Gene Symbol
MELK
Entrez Gene ID
9833
Aliases
HPK38; KIAA0175; MELK
Kinase Group
CAMK
Species
Human
PROTEIN INFORMATION
Accession #
NP_055606.1
Kinase Construct
Full Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.65
Panel
scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
26 nM
PKC-412
280 nM
VX-680/MK-0457
240 nM