MERTK
KINASE INFORMATION
Kinase Name
c-mer proto-oncogene tyrosine kinase
Entrez Gene Symbol
MERTK
Entrez Gene ID
10461
Aliases
c-mer; MER; MERTK; MGC133349; RP38
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
AAB60430.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.63
Panel
scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
32 nM
Staurosporine
6.4 nM
Sunitinib
26 nM
ZD-6474
1400 nM