MKNK2
KINASE INFORMATION
Kinase Name
MAP kinase interacting serine/threonine kinase 2
Entrez Gene Symbol
MKNK2
Entrez Gene ID
2872
Aliases
GPRK7; MKNK2; MNK2
Kinase Group
CAMK
Species
Human
PROTEIN INFORMATION
Accession #
NP_060042.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.72
Panel
scanEDGE; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
ABT-869
270 nM
AST-487
3 nM
Sorafenib
130 nM