MLK3
KINASE INFORMATION
Kinase Name
mitogen-activated protein kinase kinase kinase 11
Entrez Gene Symbol
MAP3K11
Entrez Gene ID
4296
Aliases
MAP3K11; MEKK11; MGC17114; MLK3; MLK-3; PTK1; SPRK
Kinase Group
TKL
Species
Human
PROTEIN INFORMATION
Accession #
NP_002410.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.69
Panel
Delta Set CE; Delta Set M; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CGP-52421
270 nM
PKC-412
17 nM
VX-680/MK-0457
680 nM