MST1R
KINASE INFORMATION
Kinase Name
macrophage stimulating 1 receptor (c-met-related tyrosine kinase)
Entrez Gene Symbol
MST1R
Entrez Gene ID
4486
Aliases
CD136; CDw136; MST1R; PTK8; RON
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_002438.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.72
Panel
scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
8200 nM
Staurosporine
400 nM