PAK7
KINASE INFORMATION
Kinase Name
p21 protein (Cdc42/Rac)-activated kinase 7
Entrez Gene Symbol
PAK7
Entrez Gene ID
57144
Aliases
KIAA1264; MGC26232; PAK5; PAK7
Kinase Group
STE
Species
Human
PROTEIN INFORMATION
Accession #
NP_065074.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.7
Panel
Delta Set CE; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
24 nM
Staurosporine
1.2 nM
VX-680/MK-0457
3300 nM