PCTK3
KINASE INFORMATION
Kinase Name
cyclin-dependent kinase 18
Entrez Gene Symbol
CDK18
Entrez Gene ID
5129
Aliases
CDK18; PCTAIRE; PCTAIRE3; PCTK3
Kinase Group
CMGC
Species
Human
PROTEIN INFORMATION
Accession #
NP_002587.2
Kinase Construct
Full Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.62
Panel
Delta Set CA; Delta Set CE; Delta Set I; Delta Set M; Delta Set RB; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
BMS-387032/SNS-032
44 nM
JNJ-7706621
2100 nM
Sunitinib
1700 nM