PDGFRB
KINASE INFORMATION
Kinase Name
platelet-derived growth factor receptor, beta polypeptide
Entrez Gene Symbol
PDGFRB
Entrez Gene ID
5159
Aliases
CD140B; JTK12; PDGFR; PDGFR1; PDGFRB; PDGFR-b; PDGFRbeta; PEGFR-beta
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_002600.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.63
Panel
scanEDGE; scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
28 nM
CHIR-258/TKI-258
3.8 nM
Imatinib
14 nM
MLN-518
4.5 nM
Pazopanib
2 nM
SU-14813
0.29 nM