PDPK1
KINASE INFORMATION
Kinase Name
3-phosphoinositide dependent protein kinase-1
Entrez Gene Symbol
PDPK1
Entrez Gene ID
5170
Aliases
MGC20087; MGC35290; PDK1; PDPK1; PRO0461
Kinase Group
AGC
Species
Human
PROTEIN INFORMATION
Accession #
NP_002604.1
Kinase Construct
Full Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.68
Panel
Delta Set I; scanEDGE; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
3.4 nM
CGP-52421
15 nM
LY-333531
700 nM