PIK3C2G
KINASE INFORMATION
Kinase Name
phosphoinositide-3-kinase, class 2, gamma polypeptide
Entrez Gene Symbol
PIK3C2G
Entrez Gene ID
5288
Aliases
MGC163149; PI3K-C2GAMMA; PIK3C2G
Kinase Group
Lipid
Species
Human
PROTEIN INFORMATION
Accession #
NP_004561.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.58
Panel
Delta Set CA; Delta Set CE; Delta Set I; Delta Set M; Delta Set RB; scanELECT; scanLIPID; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
230 nM
PKC-412
570 nM
Staurosporine
430 nM
Wortmannin
1500 nM