PIK3CA
KINASE INFORMATION
Kinase Name
phosphoinositide-3-kinase, catalytic, alpha polypeptide
Entrez Gene Symbol
PIK3CA
Entrez Gene ID
5290
Aliases
MGC142161; MGC142163; p110-alpha; PI3K; PIK3CA
Kinase Group
Lipid
Species
Human
PROTEIN INFORMATION
Accession #
NP_006209.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.71
Panel
Delta Set CE; Delta Set M; scanEDGE; scanELECT; scanLIPID; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
K-252a
2000 nM
PI-103
1.5 nM
Wortmannin
5.1 nM