PKAC-alpha
KINASE INFORMATION
Kinase Name
protein kinase, cAMP-dependent, catalytic, alpha
Entrez Gene Symbol
PRKACA
Entrez Gene ID
5566
Aliases
MGC102831; MGC48865; PKAa; PKACA; PKAC-a; PKACalpha; PKAC-alpha; PRKACA
Kinase Group
AGC
Species
Human
PROTEIN INFORMATION
Accession #
NP_002721.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.61
Panel
scanEDGE; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
PKC-412
720 nM
SB-202190
1700 nM
Staurosporine
19 nM