PKAC-beta
KINASE INFORMATION
Kinase Name
protein kinase, cAMP-dependent, catalytic, beta
Entrez Gene Symbol
PRKACB
Entrez Gene ID
5567
Aliases
DKFZp781I2452; MGC41879; MGC9320; PKAb; PKACB; PKAC-b; PKACbeta; PKAC-beta; PRKACB
Kinase Group
AGC
Species
Human
PROTEIN INFORMATION
Accession #
NP_002722.1
Kinase Construct
Full Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.78
Panel
Delta Set CE; Delta Set I; Delta Set M; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
AST-487
260 nM
CEP-701
160 nM
SB-202190
530 nM