PLK4
KINASE INFORMATION
Kinase Name
polo-like kinase 4 (Drosophila)
Entrez Gene Symbol
PLK4
Entrez Gene ID
10733
Aliases
PLK4; SAK; STK18
Kinase Group
Other
Species
Human
PROTEIN INFORMATION
Accession #
NP_055079.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.81
Panel
Delta Set I; Delta Set M; scanEDGE; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
1.5 nM
JNJ-7706621
120 nM
Staurosporine
0.77 nM