QSK
KINASE INFORMATION
Kinase Name
SIK family kinase 3
Entrez Gene Symbol
KIAA0999
Entrez Gene ID
23387
Aliases
FLJ12240; KIAA0999; L19; QSK; SIK3
Kinase Group
CAMK
Species
Human
PROTEIN INFORMATION
Accession #
BAA76843.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.64
Panel
Delta Set CA; Delta Set CE; Delta Set I; Delta Set M; Delta Set RB; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
120 nM
CGP-52421
230 nM
PKC-412
98 nM