RAF1
KINASE INFORMATION
Kinase Name
v-raf-1 murine leukemia viral oncogene homolog 1
Entrez Gene Symbol
RAF1
Entrez Gene ID
5894
Aliases
CRAF; c-Raf; NS5; RAF1; Raf-1
Kinase Group
TKL
Species
Human
PROTEIN INFORMATION
Accession #
NP_002871.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.68
Panel
scanEDGE; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
AMG-706
880 nM
CHIR-265/RAF-265
390 nM
Dasatinib
570 nM
Sorafenib
230 nM