RET
KINASE INFORMATION
Kinase Name
ret proto-oncogene
Entrez Gene Symbol
RET
Entrez Gene ID
5979
Aliases
CDHF12; CDHR16; HSCR1; MEN2A; MEN2B; MTC1; PTC; RET; RET51; RET-ELE1
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_065681.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.8
Panel
scanEDGE; scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
AMG-706
14 nM
CHIR-258/TKI-258
71 nM
Pazopanib
310 nM
SU-14813
37 nM
Sunitinib
12 nM
ZD-6474
34 nM