RET(V804M)
KINASE INFORMATION
Kinase Name
ret proto-oncogene
Entrez Gene Symbol
RET
Entrez Gene ID
5979
Aliases
CDHF12; CDHR16; HSCR1; MEN2A; MEN2B; MTC1; PTC; RET; RET51; RET-ELE1
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_065681.1
Kinase Construct
Partial Length
Kinase Form
Mutation (V804M)
Mutation Relevance
Activating mutation found in multiple endocrine neoplasias and familial medullary thyroid carcinomas.
Mutation References
Oncogene.
23, 6056-6063 (2004)
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.7
Panel
scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
AC220
9.1 nM
CEP-701
4.7 nM
CGP-52421
260 nM
PKC-412
20 nM
Sorafenib
22 nM
Sunitinib
5.8 nM