ROCK2
KINASE INFORMATION
Kinase Name
Rho-associated, coiled-coil containing protein kinase 2
Entrez Gene Symbol
ROCK2
Entrez Gene ID
9475
Aliases
KIAA0619; ROCK2
Kinase Group
AGC
Species
Human
PROTEIN INFORMATION
Accession #
NP_004841.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.74
Panel
scanEDGE; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
71 nM
PKC-412
2300 nM
Sunitinib
140 nM