ROS1
KINASE INFORMATION
Kinase Name
c-ros oncogene 1 , receptor tyrosine kinase
Entrez Gene Symbol
ROS1
Entrez Gene ID
6098
Aliases
c-ros-1; MCF3; ROS; ROS1
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_002935.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.7
Panel
scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
26 nM
PKC-412
430 nM
VX-680/MK-0457
610 nM