RPS6KA5(Kin.Dom.2-C-terminal)
KINASE INFORMATION
Kinase Name
ribosomal protein S6 kinase, 90kDa, polypeptide 5
Entrez Gene Symbol
RPS6KA5
Entrez Gene ID
9252
Aliases
MGC1911; MSK1; MSK1~b; MSPK1; RLPK; RPS6KA5
Kinase Group
CAMK
Species
Human
PROTEIN INFORMATION
Accession #
NP_004746.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.68
Panel
scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
960 nM
SU-14813
1500 nM
Sunitinib
1700 nM