SIK
KINASE INFORMATION
Kinase Name
salt-inducible kinase 1
Entrez Gene Symbol
SIK1
Entrez Gene ID
150094
Aliases
MSK; SIK; SIK1; SNF1LK
Kinase Group
CAMK
Species
Human
PROTEIN INFORMATION
Accession #
NP_775490.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.76
Panel
Delta Set I; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CGP-52421
66 nM
Dasatinib
3.9 nM
PKC-412
160 nM