SNARK
KINASE INFORMATION
Kinase Name
NUAK family, SNF1-like kinase, 2
Entrez Gene Symbol
NUAK2
Entrez Gene ID
81788
Aliases
DKFZp434J037; DKFZp686F01113; FLJ90349; NUAK2; SNARK
Kinase Group
CAMK
Species
Human
PROTEIN INFORMATION
Accession #
NP_112214.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.66
Panel
Delta Set CE; Delta Set I; Delta Set M; scanEDGE; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CHIR-258/TKI-258
130 nM
JNJ-7706621
26 nM
PKC-412
63 nM