SRC
KINASE INFORMATION
Kinase Name
v-src sarcoma (Schmidt-Ruppin A-2) viral oncogene homolog (avian)
Entrez Gene Symbol
SRC
Entrez Gene ID
6714
Aliases
ASV; c-SRC; p60-Src; SRC; SRC1
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_005408.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.78
Panel
scanEDGE; scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
Dasatinib
0.21 nM
VX-680/MK-0457
170 nM
ZD-6474
70 nM