SRMS
KINASE INFORMATION
Kinase Name
src-related kinase lacking C-terminal regulatory tyrosine and N-terminal myristylation sites
Entrez Gene Symbol
SRMS
Entrez Gene ID
6725
Aliases
C20orf148; dJ697K14.1; SRM; SRMS
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_543013.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.77
Panel
Delta Set M; scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
AST-487
72 nM
Dasatinib
13 nM
SU-14813
62 nM