TAK1
KINASE INFORMATION
Kinase Name
mitogen-activated protein kinase kinase kinase 7
Entrez Gene Symbol
MAP3K7
Entrez Gene ID
6885
Aliases
MAP3K7; MEKK7; TAK1; TGF1a
Kinase Group
TKL
Species
Human
PROTEIN INFORMATION
Accession #
NP_663304.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.75
Panel
scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
2.9 nM
Sorafenib
690 nM
Sunitinib
93 nM