TBK1
KINASE INFORMATION
Kinase Name
TANK-binding kinase 1
Entrez Gene Symbol
TBK1
Entrez Gene ID
29110
Aliases
FLJ11330; NAK; T2K; TBK1
Kinase Group
Other
Species
Human
PROTEIN INFORMATION
Accession #
NP_037386.1
Kinase Construct
Full Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.66
Panel
scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CGP-52421
150 nM
PKC-412
9.3 nM
Sunitinib
120 nM