TGFBR2
KINASE INFORMATION
Kinase Name
transforming growth factor, beta receptor II (70/80kDa)
Entrez Gene Symbol
TGFBR2
Entrez Gene ID
7048
Aliases
AAT3; FAA3; LDS1B; LDS2B; MFS2; RIIC; TAAD2; TGFbeta-RII; TGFBR2; TGFR-2
Kinase Group
TKL
Species
Human
PROTEIN INFORMATION
Accession #
NP_003233.4
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.67
Panel
Delta Set CA; Delta Set CE; Delta Set I; Delta Set M; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
AST-487
260 nM
CI-1033
800 nM
SB-203580
1800 nM