TRKC
KINASE INFORMATION
Kinase Name
neurotrophic tyrosine kinase, receptor, type 3
Entrez Gene Symbol
NTRK3
Entrez Gene ID
4916
Aliases
gp145(trkC); NTRK3; TRKC
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
AAA75374.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.77
Panel
Delta Set M; scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
14 nM
Sunitinib
5100 nM
VX-680/MK-0457
200 nM