TXK
KINASE INFORMATION
Kinase Name
TXK tyrosine kinase
Entrez Gene Symbol
TXK
Entrez Gene ID
7294
Aliases
BTKL; MGC22473; PSCTK5; PTK4; RLK; TKL; TXK
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_003319.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.73
Panel
scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
660 nM
CI-1033
700 nM
Dasatinib
2.1 nM