TYK2(JH1domain-catalytic)
KINASE INFORMATION
Kinase Name
tyrosine kinase 2
Entrez Gene Symbol
TYK2
Entrez Gene ID
7297
Aliases
JTK1; TYK2
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_003322.2
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.62
Panel
Delta Set M; scanEDGE; scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CP-690550
620 nM
JNJ-7706621
32 nM
PKC-412
250 nM