TYK2(JH2domain-pseudokinase)
KINASE INFORMATION
Kinase Name
tyrosine kinase 2
Entrez Gene Symbol
TYK2
Entrez Gene ID
7297
Aliases
JTK1; TYK2; Tyk2~b
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_003322.3
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.66
Panel
Delta Set M; scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
CEP-701
910 nM
Staurosporine
3100 nM
Sunitinib
360 nM