VEGFR2
KINASE INFORMATION
Kinase Name
kinase insert domain receptor (a type III receptor tyrosine kinase)
Entrez Gene Symbol
KDR
Entrez Gene ID
3791
Aliases
CD309; FLK1; FLK-1; KDR; KRD-1; Ly73; VEGFR; VEGFR2; VEGFR-2
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_002244.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Mammalian
ASSAY INFORMATION
Average Z’ Value
0.71
Panel
scanEDGE; scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
AMG-706
26 nM
CHIR-265/RAF-265
1300 nM
Pazopanib
14 nM
PTK-787
62 nM
SU-14813
2.3 nM
ZD-6474
820 nM