YES
KINASE INFORMATION
Kinase Name
v-yes-1 Yamaguchi sarcoma viral oncogene homolog 1
Entrez Gene Symbol
YES1
Entrez Gene ID
7525
Aliases
c-yes; HsT441; P61-YES; Yes; YES1
Kinase Group
TK
Species
Human
PROTEIN INFORMATION
Accession #
NP_005424.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.71
Panel
scanELECT; scanMAX; scanTK;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
Dasatinib
0.3 nM
Sunitinib
120 nM
ZD-6474
120 nM