ZAK
KINASE INFORMATION
Kinase Name
sterile alpha motif and leucine zipper containing kinase AZK
Entrez Gene Symbol
ZAK
Entrez Gene ID
51776
Aliases
AZK; MLK7; mlklak; MLT; MLTK; MRK; pk; ZAK
Kinase Group
TKL
Species
Human
PROTEIN INFORMATION
Accession #
NP_598407.1
Kinase Construct
Partial Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.75
Panel
Delta Set CA; Delta Set CE; Delta Set M; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
AMG-706
8 nM
AST-487
2.3 nM
CHIR-265/RAF-265
63 nM