p38-alpha
KINASE INFORMATION
Kinase Name
mitogen-activated protein kinase 14
Entrez Gene Symbol
MAPK14
Entrez Gene ID
1432
Aliases
CSBP1; CSBP2; CSPB1; EXIP; MAPK14; Mxi2; p38; p38a; p38ALPHA; p38-alpha; PRKM14; PRKM15; RK; SAPK2A
Kinase Group
CMGC
Species
Human
PROTEIN INFORMATION
Accession #
NP_620581.1
Kinase Construct
Full Length
Kinase Form
Wild Type
Expression System
Bacterial
ASSAY INFORMATION
Average Z’ Value
0.8
Panel
scanEDGE; scanELECT; scanMAX;
REFERENCE INHIBITOR INFORMATION
Compound
Kd
BIRB-796
0.37 nM
SB-202190
9.8 nM
SB-203580
12 nM
VX-745
2.8 nM